Prof. Dr. Olivier Baudoin

Tsitopoulou, Maria, Clemenceau, Antonin, Thesmar, Pierre, & Baudoin, Olivier. (2024). 1,4-Pd Migration-Enabled Synthesis of Fused 4-Membered Rings [Journal-article]. Journal of the American Chemical Society, 146(28), 18811–18816. https://doi.org/10.1021/jacs.4c04701

Geraci, Andrea, & Baudoin, Olivier. (2024). Fe-Catalyzed α-C(sp 3 )−H Amination of N-Heterocycles. Angewandte Chemie - International Edition. https://doi.org/10.1002/anie.202417414

Miyakoshi, Takeru, Kronenberg, Domenic, Tamaki, Sota, Lombardi, Rafael, & Baudoin, Olivier. (2024). Studies towards the Enantioselective Synthesis of Cryptowolinol via Pd⁰-Catalyzed C(sp³)-H Arylation/Parallel Kinetic Resolution. Organic Letters, null. https://doi.org/10.1021/acs.orglett.4c00386

Vyhivskyi, Oleksandr, & Baudoin, Olivier. (2024). Total Synthesis of the Diterpenes (+)-Randainin D and (+)-Barekoxide via Photoredox-Catalyzed Deoxygenative Allylation. Journal of the American Chemical Society. https://doi.org/10.1021/jacs.4c02224

Kudashev, Anton, Vergura, Stefania, Zuccarello, Marco, Bürgi, Thomas, & Baudoin, Olivier. (2023). Methylene C(sp³)−H Arylation Enables the Stereoselective Synthesis and Structure Revision of Indidene Natural Products [Journal-article]. Angewandte Chemie International Edition, 63(1). https://doi.org/10.1002/anie.202316103

Geraci, Andrea, Stojiljković, Uros, Antien, Kevin, Salameh, Nihad, & Baudoin, Olivier. (2023). Iridium(III)-Catalyzed Intermolecular C(sp³)-H Amidation for the Synthesis of Chiral 1,2-Diamines. Angewandte Chemie International Edition, 62(42), e202309263. https://doi.org/10.1002/anie.202309263

Guo, Shu-Min, Huh, Soohee, Coehlo, Max, Shen, Li, Pieters, Grégory, & Baudoin, Olivier. (2023). A C-H activation-based enantioselective synthesis of lower carbo[n]helicenes. Nature chemistry, 15, 872–880. https://doi.org/10.1038/s41557-023-01174-5

Martynova, Ekaterina A., Zuccarello, Marco, Kronenberg, Domenic, Beliš, Marek, Czapik, Agnieszka, Zhang, Ziyun, Van Hecke, Kristof, Kwit, Marcin, Baudoin, Olivier, Cavallo, Luigi, & Nolan, Steven P. (2023). Simple synthetic access to [Au(IBiox)Cl] complexes. Dalton Transactions, 52(22), 7558–7563. https://doi.org/10.1039/d3dt01357j

Salameh, Nihad, Valentini, Federica, Baudoin, Olivier, & Vaccaro, Luigi. (2023). A General Enantioselective C-H Arylation Using an Immobilized Recoverable Palladium Catalyst. ChemSusChem, 16(23). https://doi.org/10.1002/cssc.202300609

Wheatley, Matthew, Zuccarello, Marco, Tsitopoulou, Maria, Macgregor, Stuart A., & Baudoin, Olivier. (2023). Effect of α-Substitution on the Reactivity of C(sp³)-H Bonds in Pd⁰-Catalyzed C-H Arylation. ACS Catalysis, 13, 12563–12570. https://doi.org/10.1021/acscatal.3c03806

Ferlin, Francesco, Anastasiou, Ioannis, Salameh, Nihad, Miyakoshi, Takeru, Baudoin, Olivier, & Vaccaro, Luigi. (2022). C(sp³)−H Arylation Promoted by a Heterogeneous Palladium-N-Heterocyclic Carbene Complex in Batch and Continuous Flow. ChemSusChem, 15(6), e202102736. https://doi.org/10.1002/cssc.202102736

Miyakoshi, Takeru, Niggli, Nadja E., & Baudoin, Olivier. (2022). Remote Construction of N-Heterocycles via 1,4-Palladium Shift-Mediated Double C-H Activation. Angewandte Chemie International Edition, 61(17), e202116101. https://doi.org/10.1002/anie.202116101

Antien, Kevin, Geraci, Andrea, Parmentier, Michael, & Baudoin, Olivier. (2021). A New Dioxazolone for the Synthesis of 1,2-Aminoalcohols via Iridium(III)-Catalyzed C(sp; 3; )-H Amidation. Angewandte Chemie International Edition, 60(42), 22948–22955. https://doi.org/10.1002/anie.202110019

Baudoin, Olivier. (2021). A Personal Account on Industrial Collaborations in the Field of C-H Activation. Chimia, 75(11), 967–971. https://doi.org/10.2533/chimia.2021.967

Kudashev, Anton, & Baudoin, Olivier. (2021). Site-Selective Pd-Catalyzed C(sp3)-H Arylation of Heteroaromatic Ketones. Chemistry - A European Journal, 27(70), 17688–17694. https://doi.org/10.1002/chem.202103467

Melot, Romain, Zuccarello, Marco, Cavalli, Diana, Niggli, Nadja, Devereux, Michael, Bürgi, Thomas, & Baudoin, Olivier. (2021). Palladium(0)-Catalyzed Enantioselective Intramolecular Arylation of Enantiotopic Secondary C-H Bonds. Angewandte Chemie International Edition, 60(13), 7245–7250. https://doi.org/10.1002/anie.202014605

Niggli, Nadja E., & Baudoin, Olivier. (2021). Design of Chiral NHC-Carboxylates as Potential Ligands for Pd-Catalyzed Enantioselective C-H Activation. Helvetica Chimica Acta, 104(3), e2100015. https://doi.org/10.1002/hlca.202100015

Savary, David, & Baudoin, Olivier. (2021). Enantioselective Pd0-Catalyzed C(sp2)-H Arylation for the Synthesis of Chiral Warped Molecules. Angewandte Chemie International Edition, 10. https://doi.org/10.1002/anie.202013303

Vyhivskyi, Oleksandr, Kudashev, Anton, Miyakoshi, Takeru, & Baudoin, Olivier. (2021). Chiral Catalysts for Pd-0-Catalyzed Enantioselective C-H Activation. Chemistry - A European Journal, 27(4), 1231–1257. https://doi.org/10.1002/chem.202003225

Baudoin, Olivier. (2020). Multiple Catalytic C-H Bond Functionalization for Natural Product Synthesis. Angewandte Chemie (International ed. in English), 10. https://doi.org/10.1002/anie.202001224

Baumgartner, Yann, & Baudoin, Olivier. (2020). One-Pot Alkene Hydroboration/Palladium-Catalyzed Migratory Suzuki−Miyaura Cross-Coupling. ACS Catalysis, 10, 10508–10515. https://doi.org/10.1021/acscatal.0c02755

Carny, Tomas, Rocaboy, Ronan, Clemenceau, Antonin, & Baudoin, Olivier. (2020). Synthesis of Amides and Esters by Palladium(0)-Catalyzed Carbonylative C(sp3)-H Activation. Angewandte Chemie International Edition, 59(43), 18980–18984. https://doi.org/10.1002/anie.202007922

Clemenceau, Antonin, Thesmar, Pierre, Gicquel, Maxime, Le Flohic, Alexandre, & Baudoin, Olivier. (2020). Direct Synthesis of Cyclopropanes from gem-Dialkyl Groups through Double C-H Activation. Journal of the American Chemical Society, 142(36), 15355–15361. https://doi.org/10.1021/jacs.0c05887

Nguyen, Qui-Hien, Guo, Shu-Min, Royal, Titouan, Baudoin, Olivier, & Cramer, Nicolai. (2020). Intermolecular Palladium(0)-Catalyzed Atropo-enantioselective C-H Arylation of Heteroarenes. Journal of American Chemical Society, 142(5), 2161–2167. https://doi.org/10.1021/jacs.9b12299

Thesmar, Pierre, Coomar, Seemon, Prescimone, Alessandro, Häussinger, Daniel, Gillingham, Dennis, & Baudoin, Olivier. (2020). Divergent Synthesis of Bioactive Dithiodiketopiperazine Natural Products Based on a Double C(sp3)−H Activation Strategy. Chemistry - A European Journal, 26. https://doi.org/10.1002/chem.202003683

Lin, Weilong, Zhang, Ke-Feng, & Baudoin, Olivier. (2019). Regiodivergent enantioselective C-H functionalization of Boc-1,3-oxazinanes for the synthesis of beta(2)- and beta(3)-amino acids. Nature Catalysis, 2(10), 882–888. https://doi.org/10.1038/s41929-019-0336-1

Melot, Romain, Craveiro, Marcus V., & Baudoin, Olivier. (2019). Total Synthesis of (Nor)illudalane Sesquiterpenes Based on a C(sp3)-H Activation Strategy. Journal of Organic Chemistry, 84(20), 12933–12945. https://doi.org/10.1021/acs.joc.9b01669

Melot, Romain, Craveiro, Marcus V., Burgi, Thomas, & Baudoin, Olivier. (2019). Divergent Enantioselective Synthesis of (Nor)illudalane Sesquiterpenes via Pd-0-Catalyzed Asymmetric C(sp(3))-H Activation. Organic Letters, 21(3), 812–815. https://doi.org/10.1021/acs.orglett.8b04086

Rocaboy, Ronan, Anastasiou, Ioannis, & Baudoin, Olivier. (2019). Redox-Neutral Coupling between Two C(sp3)-H Bonds Enabled by 1,4-Palladium Shift for the Synthesis of Fused Heterocycles. Angewandte Chemie International Edition, 58(41), 14625–14628. https://doi.org/10.1002/anie.201908460

Rocaboy, Ronan, & Baudoin, Olivier. (2019). 1,4-Palladium Shift/C(sp(3))-H Activation Strategy for the Remote Construction of Five-Membered Rings. Organic Letters, 21(5), 1434–1437. https://doi.org/10.1021/acs.orglett.9b00187

Royal, Titouan, & Baudoin, Olivier. (2019). Pd-catalyzed gamma-arylation of gamma,delta-unsaturated O-carbamates via an unusual haptotropic rearrangement. Chemical Science, 10(8), 2331–2335. https://doi.org/10.1039/c8sc05058a

Thesmar, Pierre, & Baudoin, Olivier. (2019). Efficient and Divergent Total Synthesis of (-)-Epicoccin G and (-)-Rostratin A Enabled by Double C(sp; 3; )-H Activation. Journal of the American Chemical Society, 141, 15779–15783. https://doi.org/10.1021/jacs.9b09359

Rocaboy, Ronan, Dailler, David, & Baudoin, Olivier. (2018). A Four-Step Synthesis of (±)-γ-Lycorane via Pd0-Catalyzed Double C(sp2)-H/C(sp3)-H Arylation. Organic Letters, 20(3), 772–775. https://doi.org/10.1021/acs.orglett.7b03909

Rocaboy, Ronan, Dailler, David, Zellweger, Florian, Neuburger, Markus, Salomé, Christophe, Clot, Eric, & Baudoin, Olivier. (2018). Domino Pd0-Catalyzed C(sp3)-H Arylation/Electrocyclic Reactions via Benzazetidine Intermediates. Angewandte Chemie International Edition, 57(37), 12131–12135. https://doi.org/10.1002/anie.201807097

Yang, Lei, Neuburger, Markus, & Baudoin, Olivier. (2018). Chiral Bifunctional Phosphine-Carboxylate Ligands for Palladium(0)-Catalyzed Enantioselective C-H Arylation. Angewandte Chemie International Edition, 57(5), 1394–1398. https://doi.org/10.1002/anie.201712061

Zhang, Ke-Feng, Christoffel, Fadri, & Baudoin, Olivier. (2018). Barbier-Negishi Coupling of Secondary Alkyl Bromides with Aryl and Alkenyl Triflates and Nonaflates. Angewandte Chemie International Edition, 57(7), 1982–1986. https://doi.org/10.1002/anie.201711990

Baudoin, Olivier. (2017). Ring Construction by Palladium(0)-Catalyzed C(sp(3))-H Activation. Accounts of Chemical Research, 50(4), 1114–1123. https://doi.org/10.1021/acs.accounts.7b00099

Dailler, David, Rocaboy, Ronan, & Baudoin, Olivier. (2017). Synthesis of β-Lactams by Palladium(0)-Catalyzed C(sp3)−H Carbamoylation. Angewandte Chemie International Edition, 56(25), 7218–7222. https://doi.org/10.1002/anie.201703109

Goutierre, Anne-Sophie, Trinh, Huu Vinh, Larini, Paolo, Jazzar, Rodolphe, & Baudoin, Olivier. (2017). Comparative Structural Analysis of Biarylphosphine Ligands in Arylpalladium Bromide and Malonate Complexes. Organometallics, 36(1), 129–135. https://doi.org/10.1021/acs.organomet.6b00535

Holstein, Philipp M., Holstein, Julian J., Escudero-Adan, Eduardo C., Baudoin, Olivier, & Echavarren, Antonio M. (2017). Ferrocene derivatives of liquid chiral molecules allow assignment of absolute configuration by X-ray crystallography. Tetrahedron: Asymmetry, 28(10), 1321–1329. https://doi.org/10.1016/j.tetasy.2017.09.002

Royal, Titouan, Baumgartner, Yann, & Baudoin, Olivier. (2017). Enantioselective α-Arylation of O-Carbamates via Sparteine-Mediated Lithiation and Negishi Cross-Coupling. Organic Letters, 19(1), 166–169. https://doi.org/10.1021/acs.orglett.6b03472

Yang, Lei, Melot, Romain, Neuburger, Markus, & Baudoin, Olivier. (2017). Palladium(0)-catalyzed asymmetric C(sp3)-H arylation using a chiral binol-derived phosphate and an achiral ligand. Chemical Science, 8(2), 1344–1349. https://doi.org/10.1039/c6sc04006c

Holstein, P. M., Dailler, D., Vantourout, J., Shaya, J., Millet, A., & Baudoin, O. (2016). Synthesis of Strained γ-Lactams by Palladium(0)-Catalyzed C(sp3)-H Alkenylation and Application to Alkaloid Synthesis. Angewandte Chemie - International Edition, 55(8), 2805–2809. https://doi.org/10.1002/anie.201511457

Baudoin, Olivier. (2016). Selectivity Control in the Palladium-catalyzed Cross-coupling of Alkyl Nucleophiles. Chimia, 70(11), 768–772. https://doi.org/10.2533/chimia.2016.768

Dupuy, Stéphanie, Zhang, Ke-Feng, Goutierre, Anne-Sophie, & Baudoin, Olivier. (2016). Terminal-Selective Functionalization of Alkyl Chains by Regioconvergent Cross-Coupling. Angewandte Chemie International Edition, 55(47), 14793–14797. https://doi.org/10.1002/anie.201608535

Holstein, Philipp M., Dailler, David, Vantourout, Julien, Shaya, Janah, Millet, Anthony, & Baudoin, Olivier. (2016). Synthesis of Strained γ-Lactams by Palladium(0)-Catalyzed C(sp3)−H Alkenylation and Application to Alkaloid Synthesis. Angewandte Chemie, 128(8), 2855–2859. https://doi.org/10.1002/ange.201511457

Martin, Anthony, Vors, Jean-Pierre, & Baudoin, Olivier. (2016). Synthesis of Conformationally Constrained Esters and Amines by Pd-Catalyzed α-Arylation of Hindered Substrates. ACS Catalysis, 6(6), 3941–3945. https://doi.org/10.1021/acscatal.6b00943

Millet, A., & Baudoin, O. (2016). Palladium-catalyzed β-Selective C(sp3)-H arylation of N-boc-piperidines. Organic Syntheses, 92, 76–90. https://doi.org/10.15227/orgsyn.92.0076

Prieto, Alexis, Baudoin, Olivier, Bouyssi, Didier, & Monteiro, Nuno. (2016). Electrophilic trifluoromethylation of carbonyl compounds and their nitrogen derivatives under copper catalysis. Chemical Communications, 52(5), 869–881. https://doi.org/10.1039/c5cc05954b

Dailler, David, Danoun, Grégory, & Baudoin, Olivier. (2016). Applications of Catalytic Organometallic C(sp3)-H Bond Functionalization. In Dix-neuf, Pierre H.; Doucet, Henri (ed.), C-H bond activation and catalytic functionalization II (pp. 133–154). Springer International Publishing. https://doi.org/10.1007/3418_2015_122

Prieto, A., Landart, M., Baudoin, O., Monteiro, N., & Bouyssi, D. (2015). Copper-Catalyzed Trifluoromethylation of Aliphatic N-Arylhydrazones: A Concise Synthetic Entry to 2-Trifluoromethylindoles from Simple Aldehydes. Advanced Synthesis and Catalysis, 357(13), 2939–2943. https://doi.org/10.1002/adsc.201500237

Holstein, P. M., Vogler, M., Larini, P., Pilet, G., Clot, E., & Baudoin, O. (2015). Efficient Pd0-Catalyzed Asymmetric Activation of Primary and Secondary C-H Bonds Enabled by Modular Binepine Ligands and Carbonate Bases. ACS Catalysis, 5(7), 4300–4308. https://doi.org/10.1021/acscatal.5b00898

Dailler, D., Danoun, G., Ourri, B., & Baudoin, O. (2015). Divergent Synthesis of Aeruginosins Based on a C(sp3)£H Activation Strategy. Chemistry - A European Journal, 21(26), 9370–9379. https://doi.org/10.1002/chem.201501370

Dailler, D., Danoun, G., & Baudoin, O. (2015). A General and Scalable Synthesis of Aeruginosin Marine Natural Products Based on Two Strategic C(sp3)-H Activation Reactions. Angewandte Chemie - International Edition, 54(16), 4919–4922. https://doi.org/10.1002/anie.201500066

Kefalidis, C. E., Davi, M., Holstein, P. M., Clot, E., & Baudoin, O. (2014). Mechanistic study of the selectivity of olefin versus cyclobutene formation by palladium(0)-catalyzed intramolecular C(sp3)-H activation. Journal of Organic Chemistry, 79(24), 11903–11910. https://doi.org/10.1021/jo501610x

Nella, N., Parker, E., Hitce, J., Larini, P., Jazzar, R., & Baudoin, O. (2014). Efficient Pd-Catalyzed Allene Synthesis from Alkynes and Aryl Bromides through an Intramolecular Base-Assisted Deprotonation (iBAD) Mechanism. Chemistry - A European Journal, 20(41), 13272–13278. https://doi.org/10.1002/chem.201403213

Prieto, A., Jeamet, E., Monteiro, N., Bouyssi, D., & Baudoin, O. (2014). Copper-catalyzed β-trifluoromethylation of conjugated hydrazones. Organic Letters, 16(18), 4770–4773. https://doi.org/10.1021/ol5022228

Janody, S., Jazzar, R., Comte, A., Holstein, P. M., Vors, J.-P., Ford, M. J., & Baudoin, O. (2014). Synthesis of 1-indanols and 1-indanamines by intramolecular palladium(0)-catalyzed C(sp3)-H arylation: Impact of conformational effects. Chemistry - A European Journal, 20(35), 11084–11090. https://doi.org/10.1002/chem.201402907

Millet, A., & Baudoin, O. (2014). Palladium-catalyzed γ-selective arylation of zincated Boc-allylamines. Organic Letters, 16(15), 3998–4000. https://doi.org/10.1021/ol5018257

Millet, A., Dailler, D., Larini, P., & Baudoin, O. (2014). Ligand-controlled α- And β-arylation of acyclic N-boc amines. Angewandte Chemie - International Edition, 53(10), 2678–2682. https://doi.org/10.1002/anie.201310904

Davi, M., Comte, A., Jazzar, R., & Baudoin, O. (2014). Synthesis of Cyclobutarenes by Palladium‐Catalyzed C (sp 3 )‐ H Bond Arylation: Preparation of Methyl 7‐Methylbicyclo[4.2.0]Octa‐1,3,5‐Triene‐7‐Carboxylate (Other) [Other, Wiley]. 510–518. https://doi.org/10.1002/0471264229.os089.49

Aspin, S., López-Suárez, L., Larini, P., Goutierre, A.-S., Jazzar, R., & Baudoin, O. (2013). Palladium-catalyzed β-arylation of silyl ketene acetals and application to the synthesis of benzo-fused δ-lactones. Organic Letters, 15(19), 5056–5059. https://doi.org/10.1021/ol402398s

Pierre, C., & Baudoin, O. (2013). Intramolecular PdII-catalyzed dehydrogenative C(sp 3)-C(sp2) coupling: An alternative to Pd 0-catalyzed C(sp3)-H arylation from aryl halides? Tetrahedron, 69(22), 4473–4478. https://doi.org/10.1016/j.tet.2012.11.060

Pair, E., Monteiro, N., Bouyssi, D., & Baudoin, O. (2013). Copper-catalyzed trifluoromethylation of N,N-dialkylhydrazones. Angewandte Chemie - International Edition, 52(20), 5346–5349. https://doi.org/10.1002/anie.201300782

Millet, A., Larini, P., Clot, E., & Baudoin, O. (2013). Ligand-controlled β-selective C(sp3)-H arylation of N-Boc-piperidines. Chemical Science, 4(5), 2241–2247. https://doi.org/10.1039/c3sc50428j

Aspin, S., Goutierre, A.-S., Larini, P., Jazzar, R., & Baudoin, O. (2012). Synthesis of aromatic α-aminoesters: Palladium-catalyzed long-range arylation of primary Csp3-H bonds. Angewandte Chemie - International Edition, 51(43), 10808–10811. https://doi.org/10.1002/anie.201206237

Sofack-Kreutzer, J., Martin, N., Renaudat, A., Jazzar, R., & Baudoin, O. (2012). Synthesis of hexahydroindoles by intramolecular C sp 3-H alkenylation: Application to the synthesis of the core of aeruginosins. Angewandte Chemie - International Edition, 51(41), 10399–10402. https://doi.org/10.1002/anie.201205403

Martin, N., Pierre, C., Davi, M., Jazzar, R., & Baudoin, O. (2012). Diastereo- and enantioselective intramolecular C(sp3)-H arylation for the synthesis of fused cyclopentanes. Chemistry - A European Journal, 18(15), 4480–4484. https://doi.org/10.1002/chem.201200018

Larini, P., Kefalidis, C. E., Jazzar, R., Renaudat, A., Clot, E., & Baudoin, O. (2012). On the mechanism of the palladium-catalyzed β-arylation of ester enolates. Chemistry - A European Journal, 18(7), 1932–1944. https://doi.org/10.1002/chem.201103153

Guyonnet, M., & Baudoin, O. (2012). Synthesis of tricyclic nitrogen heterocycles by a sequence of palladium-catalyzed N-H and C(sp 3)-H arylations. Organic Letters, 14(1), 398–401. https://doi.org/10.1021/ol2031763

Baudoin, O. (2011). Transition metal-catalyzed arylation of unactivated C(sp3)–H bonds. Chemical Society Reviews, 40(10), 4902–4911. https://doi.org/10.1039/c1cs15058h

Pierre, C., & Baudoin, O. (2011). Synthesis of polycyclic molecules by double C(sp2)-H/C(sp 3)-H arylations with a single palladium catalyst. Organic Letters, 13(7), 1816–1819. https://doi.org/10.1021/ol200329e

Kefalidis, C. E., Baudoin, O., & Clot, E. (2010). DFT study of the mechanism of benzocyclobutene formation by palladium-catalysed C(sp3)-H activation: Role of the nature of the base and the phosphine. 39, 10528–10535. https://doi.org/10.1039/c0dt00578a

Renaudat, A., Jean-GÚrard, L., Jazzar, R., Kefalidis, C. E., Clot, E., & Baudoin, O. (2010). Palladium-catalyzed β arylation of carboxylic esters. Angewandte Chemie - International Edition, 49(40), 7261–7265. https://doi.org/10.1002/anie.201003544

Rousseaux, S., Davi, M., Sofack-Kreutzer, J., Pierre, C., Kefalidis, C. E., Clot, E., Fagnou, K., & Baudoin, O. (2010). Intramolecular palladium-catalyzed alkane C-H arylation from aryl chlorides. Journal of the American Chemical Society, 132(31), 10706–10716. https://doi.org/10.1021/ja1048847

Colombel, V., Joncour, A., Thoret, S., Dubois, J., Bignon, J., Wdzieczak-Bakala, J., & Baudoin, O. (2010). Synthesis of antimicrotubule dibenzoxepines. Tetrahedron Letters, 51(23), 3127–3129. https://doi.org/10.1016/j.tetlet.2010.04.039

Jazzar, R., Hitce, J., Renaudat, A., Sofack-Kreutzer, J., & Baudoin, O. (2010). Functionalization of organic molecules by transition-metal-catalyzed C(sp3)-H activation. Chemistry - A European Journal, 16(9), 2654–2672. https://doi.org/10.1002/chem.200902374

Colombel, V., & Baudoin, O. (2009). Synthetic approaches to amino analogues of N-acetylcolchinol. Journal of Organic Chemistry, 74(11), 4329–4335. https://doi.org/10.1021/jo900632a

Chaumontet, M., Retailleau, P., & Baudoin, O. (2009). Cycloadditions of 1,1-disubstituted benzocyclobutenes obtained by C(sp 3)-H activation. Journal of Organic Chemistry, 74(4), 1774–1776. https://doi.org/10.1021/jo802471u

Chaumontet, M., Piccardi, R., & Baudoin, O. (2009). Synthesis of 3,4-dihydroisoquinolines by a C(sp3)-H activation/electrocyclization strategy: Total synthesis of coralydine. Angewandte Chemie - International Edition, 48(1), 179–182. https://doi.org/10.1002/anie.200804444

Joncour, A., Liu, J.-M., Décor, A., Thoret, S., Wdzieczak-Bakala, J., Bignon, J., & Baudoin, O. (2008). Synthesis of anti-microtubule biaryls and preliminary evaluation as vascular-disrupting agents. ChemMedChem, 3(11), 1731–1739. https://doi.org/10.1002/cmdc.200800181

Chaumontet, M., Piccardi, R., Audic, N., Hitce, J., Peglion, J.-L., Clot, E., & Baudoin, O. (2008). Synthesis of benzocyclobutenes by palladium-catalyzed C-H activation of methyl groups: Method and mechanistic study. Journal of the American Chemical Society, 130(45), 15157–15166. https://doi.org/10.1021/ja805598s

Baudoin, O. (2008). Synthesis of tubulin-binding bridged biaryls via intermolecular Suzuki coupling. Comptes Rendus Chimie, 11(1-2), 38–42. https://doi.org/10.1016/j.crci.2007.02.016

Joncour, A., Décor, A., Liu, J.-M., Tran Huu Dau, M.-E., & Baudoin, O. (2007). Asymmetric synthesis of antimicrotubule biaryl hybrids of allocolchicine and steganacin. Chemistry - A European Journal, 13(19), 5450–5465. https://doi.org/10.1002/chem.200601764

Baudoin, O. (2007). New approaches for decarboxylative biaryl coupling. Angewandte Chemie - International Edition, 46(9), 1373–1375. https://doi.org/10.1002/anie.200604494

Hitce, J., Retailleau, P., & Baudoin, O. (2007). Palladium-catalyzed intramolecular C(sp3)-H functionalization: Catalyst development and synthetic applications. Chemistry - A European Journal, 13(3), 792–799. https://doi.org/10.1002/chem.200600811

Bonneau, A.-L., Robert, N., Hoarau, C., Baudoin, O., & Marsais, F. (2007). A new synthetic approach to biaryls of the rhazinilam type. Application to synthesis of three novel phenylpyridine-carbamate analogues. Organic and Biomolecular Chemistry, 5(1), 175–183. https://doi.org/10.1039/b613173e

Hitce, J., & Baudoin, O. (2007). Substituted benzocarbocycles by palladium-catalyzed cascade reactions featuring a C(sp3) - H activation step. Advanced Synthesis and Catalysis, 349(11-12), 2054–2060. https://doi.org/10.1002/adsc.200700099

Joncour, A., Décor, A., Thoret, S., Chiaroni, A., & Baudoin, O. (2006). Biaryl axis as a stereochemical relay for the enantioselective synthesis of antimicrotubule agents. Angewandte Chemie - International Edition, 45(25), 4149–4152. https://doi.org/10.1002/anie.200600451

Décor, A., Monse, B., Martin, M.-T., Chiaroni, A., Thoret, S., Guénard, D., Guéritte, F., & Baudoin, O. (2006). Synthesis and biological evaluation of B-ring analogues of (-)-rhazinilam. Bioorganic and Medicinal Chemistry, 14(7), 2314–2332. https://doi.org/10.1016/j.bmc.2005.11.011

Décor, A., Bellocq, D., Thoison, O., Lekieffre, N., Chiaroni, A., Ouazzani, J., Cresteil, T., Guéritte, F., & Baudoin, O. (2006). In vitro oxidative metabolism study of (-)-rhazinilam. Bioorganic and Medicinal Chemistry, 14(5), 1558–1564. https://doi.org/10.1016/j.bmc.2005.10.015

Baudoin, O. (2005). The asymmetric Suzuki coupling route to axially chiral biaryls. European Journal of Organic Chemistry, 20, 4223–4229. https://doi.org/10.1002/ejoc.200500394

Ding, H., Lu, W., Li, H., Yang, L., Zhang, Q., Zhou, C., Wu, X., Baudoin, O., Cai, J., Guéritte, F., & Zhao, Y. (2005). Synthesis and biological evaluation of novel compounds related to 1-arylnaphthalene lignans and isoquinolines. Chemistry and Biodiversity, 2(9), 1217–1231. https://doi.org/10.1002/cbdv.200590092

Baudoin, O., Guenard, D., & Gueritte, F. (2004). The Chemistry and Biology of Rhazinilam and Analogues [Journal-article]. Mini-Reviews in Organic Chemistry, 1(3), 333–341. https://doi.org/10.2174/1570193043403226

Baudoin, O., Herrbach, A., & Guéritte, F. (2003). The Palladium-Catalyzed C-H Activation of Benzylic gem-Dialkyl Groups. Angewandte Chemie - International Edition, 42(46), 5736–5740. https://doi.org/10.1002/anie.200352461

Herrbach, A., Marinetti, A., Baudoin, O., Guénard, D., & Guéritte, F. (2003). Asymmetric synthesis of an axially chiral antimitotic biaryl via an atropo-enantioselective Suzuki cross-coupling. Journal of Organic Chemistry, 68(12), 4897–4905. https://doi.org/10.1021/jo034298y

Baudoin, O., Décor, A., Cesario, M., & Guéritte, F. (2003). A Novel 1,3-Central-to-Axial Chirality Induction Approach to Cyclooctadiene Lignans. Synlett, 13, 2009–2012. https://doi.org/10.1055/s-2003-42039

Baudoin, O., Claveau, F., Thoret, S., Herrbach, A., Guénard, D., & Guéritte, F. (2002). Synthesis and biological evaluation of A-ring biaryl-carbamate analogues of rhazinilam. Bioorganic and Medicinal Chemistry, 10(11), 3395–3400. https://doi.org/10.1016/S0968-0896(02)00270-5

Baudoin, O., Cesario, M., Guénard, D., & Guéritte, F. (2002). Application of the palladium-catalyzed borylation/Suzuki coupling (BSC) reaction to the synthesis of biologically active biaryl lactams. Journal of Organic Chemistry, 67(4), 1199–1207. https://doi.org/10.1021/jo0160726

Baudoin, O., Guénard, D., & Guéritte, F. (2000). Palladium-catalyzed borylation of ortho-substituted phenyl halides and application to the one-pot synthesis of 2,2′-disubstituted biphenyls. Journal of Organic Chemistry, 65(26), 9268–9271. https://doi.org/10.1021/jo005663d